Kubudirira uye basa repaclitaxel

Paclitaxel inobva kuTaxus chinensis uye ndicho chinhu chekutanga kuwanikwa chiine inhibitory mhedzisiro pamasero ebundu.Chimiro che paclitaxel chakaoma, uye mashandisirwo ayo ekurapa anonyanya kuratidzwa mukurapa kenza yemazamu, kenza yemapapu, uye ovarian cancer.Paclitaxelndeyechipiri metabolite yakatorwa kubva kugwati reTaxus chinensis neAmerican chemist, ine yakanaka anti-tumor athari.Ngatitarisei kushanda uye basa repaclitaxel.

Kubudirira uye basa repaclitaxel

Kubudirira uye basa repaclitaxel

1. Anti-tumor effect

Paclitaxel is anti-microtubule antitumor drug.Paclitaxel inogona kusimudzira microtubule kusangana nekusimudzira polymerization yespinosomal tubulin subunits, kunyangwe muyananisi anodiwa kune yakajairika microtubule musangano (seGTP, guanosine triphosphate, nezvimwewo)., etc.) inogonawo kuva nemigumisiro iyi, zvichiita kuti pave nekuumbwa kwezvisina kushanda, zvakagadzikana microtubules.

2. Anti-cancer effect

Paclitaxel ine anticancer mhedzisiro pane yakashata sarcoma cell mitsara, leukemia uye yakaipa melanoma.Paclitaxel zvakare mushonga wekutanga-mutsetse wevakadzi vane advanced mazamu uye ovarian cancer.Paclitaxel inogona kusunga kune microtubules, iyo inogona "kuomesa" uye kudzivirira kupatsanurwa kwemakromosomes panguva yekuparadzaniswa kwesero, iyo inogona kukurumidza kuuraya masero ekenza.

3. Kurapa kwe rheumatoid arthritis

Zvidzidzo zvakaratidza kuti paclitaxel yakabvumidzwa neFDA pakurapa rheumatoid arthritis, uye paclitaxel gel inogadzirwa nemusoro.paclitaxel yekurapa rheumatoid arthritis.

Ongorora: Iko kugona kushanda uye mashandisirwo anotsanangurwa muchinyorwa chino anotorwa kubva kumabhuku akaburitswa.

paclitaxel API

Kuwedzera kuverenga:Yunnan Hande Biotechnology Co., Ltd yanga yakatarisana nekugadzirwa kwepaclitaxel kwemakore makumi maviri nemasere.Ndiyo yekutanga yakazvimirira kugadzira pasi rose-yakagadzirwa anticancer drug paclitaxel iyo yakatenderwa neUS FDA, European EDQM, Australian TGA, China CFDA, India, Japan nemamwe masangano anodzora nyika.enterprise.Kana uchida kutengaPurogiramu inonzi Paclitaxel,ndapota taura nesu online.


Nguva yekutumira: Sep-30-2022